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Gabexate mesylate
CAS No. 56974-61-9
Gabexate mesylate( —— )
Catalog No. M15075 CAS No. 56974-61-9
Gabexate Mesylate is a Factor X inhibitor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 46 | In Stock |
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| 10MG | 74 | In Stock |
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| 25MG | 122 | In Stock |
|
| 50MG | 178 | In Stock |
|
| 100MG | 291 | In Stock |
|
| 200MG | 379 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameGabexate mesylate
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NoteResearch use only, not for human use.
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Brief DescriptionGabexate Mesylate is a Factor X inhibitor.
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DescriptionGabexate Mesylate is a Factor X inhibitor.
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In VitroCell Proliferation Assay Cell Line:HepG2 cells Concentration:100, 300, and 1000 μM Incubation Time:72 hours Result:The proliferation rate decreased in a dose-dependent manner.
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In VivoAnimal Model:Male Sprague-Dawley rats (100-120 g) with spinal nerve ligation (SNL) Dosage:20 mg/kg Administration:Intraperitoneally; daily; from 3rd day until the 14th day Result:Showed a higher PWT than those of the vehicle-treated group. Markedly decreased the expression of p65. Attenuated the expressions of IL-1, IL-6, and TNF-α at 7th day.
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Synonyms——
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PathwayProteasome/Ubiquitin
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TargetSerine Protease
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RecptorSerine Protease
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Research AreaCardiovascular Disease
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Indication——
Chemical Information
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CAS Number56974-61-9
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Formula Weight417.48
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Molecular FormulaC17H27N3O7
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Purity>98% (HPLC)
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SolubilityEthanol: 83 mg/mL (198.81 mM); Water: 12 mg/mL (28.74 mM); DMSO: 83 mg/mL (198.81 mM)
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SMILESCS(O)(=O)=O.CCOC(=O)C1=CC=C(OC(=O)CCCCCN=C(N)N)C=C1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Erba F, et al. Biochem Pharmacol. 2001 Feb 1;61(3):271-6.
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